論文 - 大金 賢司
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In-gel refolding allows fluorescence detection of fully denatured GFPs after SDS-PAGE
Analytical Biochemistry, Elsevier, 702巻(頁115861), 2025年04月, Misa Shiratori, Rio Tsuyuki, Miwako Asanuma, Saki Kawabata, Hiromasa Yoshioka, Kenji Ohgane, 原著, 研究論文(学術雑誌), 第一著者相当
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Synthesis and Biological Assessment of Eucalyptin: Magic Methyl Effects
International Journal of Molecular Sciences, MDPI, 26巻7号(頁3391 - ), 2025年04月, Kanta Fuchiyama, Yuka Yabuki, Yuzu Yamamoto, Ryuki Asakawa, Saki Matsumoto, Yuuka Ibayashi, yuuki furuyama, Kenji Ohgane, Shinji Kamisuki, Koichi Watashi, Makoto Matsubayashi, Kouji Kuramochi, 原著, 研究論文(学術雑誌), 共著者
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Clozapine as an E3 Ligand for PROTAC Technology
ACS Medicinal Chemistry Letters, , 16巻2号(頁258 - 262), 2025年02月, Reina Takano, Nobumichi Ohoka, Takashi Kurohara, Noriaki Arakawa, Kenji Ohgane, Takao Inoue, Hidetomo Yokoo, Yosuke Demizu, 原著, 研究論文(学術雑誌), 共著者
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Phenylboronic acids as pH-selective ligands for arylsulfatase B: a lead for pharmacological chaperones against Maroteaux–Lamy syndrome
chemRxiv, American Chemical Society (ACS), 2025年01月, Fumika Karaki, Kyoko Hidaka, Yuko Nishiyama, Ami Taniguchi, Yuichi Hashimoto, Kenji Ohgane, Hideaki Fujii, 原著, 研究論文(学術雑誌), 第一著者相当
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In-gel refolding allows fluorescence detection of fully denatured GFPs after SDS-PAGE
bioRxiv, , 2024年10月, Misa Shiratori, Rio Tsuyuki, Miwako Asanuma, Saki Kawabata, Hiromasa Yoshioka, Kenji Ohgane, 原著, 研究論文(学術雑誌), 第一著者相当
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Plakevulin A induces apoptosis and suppresses IL-6-induced STAT3 activation in HL60 cells.
Bioorganic & medicinal chemistry letters, , 110巻(頁129886 - ), 2024年09月, Misaki Kabasawa, Masateru Furuta, Yuuka Ibayashi, Kaori Kanemaru, Haruki Kohatsu, Fumiyo Kuramochi, Kenji Yamatoya, Kazuya Nakata, Yoshikazu Nakamura, Shusuke Tomoshige, Kenji Ohgane, Yuuki Furuyama, Ryoko Takasawa, Susumu Kobayashi, Fumio Sugawara, Masahiko Ikekita, Kouji Kuramochi, 原著, 研究論文(学術雑誌), 共著者
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Mutant induced neurons and humanized mice enable identification of Niemann-Pick type C1 proteostatic therapies
JCI Insight, , 9巻20号(頁e179525 - ), 2024年08月, Ruth D. Azaria, Adele B. Correia, Kylie J. Schache, Manuela Zapata, Koralege C. Pathmasiri, Varshasnata Mohanty, Dharma T. Nannapaneni, Brandon L. Ashfeld, Paul Helquist, Olaf Wiest, Kenji Ohgane, Qingqing Li, Ross A. Fredenburg, Brian S.J. Blagg, Stephanie M. Cologna, Mark L. Schultz, Andrew P. Lieberman, 原著, 研究論文(学術雑誌), 共著者
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A small-molecule degron with a phenylpropionic acid scaffold
Bioorganic & Medicinal Chemistry, Elsevier, 109巻(頁117789 - ), 2024年07月, Shusuke Tomoshige, Fumiko Komatsu, Tomoko Kikuchi, Miku Sugiyama, Yushi Kawasaki, Kenji Ohgane, Yuuki Furuyama, Shinichi Sato, Minoru Ishikawa, Kouji Kuramochi, 原著, 研究論文(学術雑誌), 共著者
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Anti-hepatitis C Virus Activity of Juglorubin Derivatives
Chem Pharm Bull, , 71巻11号(頁843 - 845), 2023年11月, OHASHI Hirofumi, NISHIOKA Kazane, KURIHARA Tomoki, NAKAMURA Kou, YAMASAKI Masako, IBAYASHI Yuuka, FUCHIYAMA Kanta, KAMO Shogo, FURUYAMA Yuuki, OHGANE Kenji, OKADA Maiko, KAMISUKI Shinji, WATASHI Koichi, KURAMOCHI Kouji, 原著, 研究論文(学術雑誌), 共著者
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Lysine long-chain fatty acylation regulates the TEAD transcription factor.
Cell reports, Cell Press, 42巻4号(頁112388 - ), 2023年04月, Kota Noritsugu, Takehiro Suzuki, Kosuke Dodo, Kenji Ohgane, Yasue Ichikawa, Kota Koike, Satoshi Morita, Takashi Umehara, Kenji Ogawa, Mikiko Sodeoka, Naoshi Dohmae, Minoru Yoshida, Akihiro Ito, 原著, 研究論文(学術雑誌), 共著者
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Fine-tuning of nitrogen-containing bisphosphonate esters that potently induce degradation of HMG-CoA reductase
Bioorganic & Medicinal Chemistry, Elsevier, 78巻(頁117145 - ), 2022年12月, Kota Kawamura, Hiromasa Yoshioka, Chikako Sato, Tomoko Yajima, Yuuki Furuyama, Kouji Kuramochi, Kenji Ohgane, 原著, 研究論文(学術雑誌), 第一著者相当
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Synthesis and cytotoxic activities of 8- and 6-demethyleucalyptins
Bioscience, Biotechnology, and Biochemistry, , 86巻9号(頁1200 - 1206), 2022年08月, ASAKAWA Ryuki, FUCHIYAMA Kanta, ISHII Yunosuke, HOSAKA Keisuke, KOBAYASHI Atsushi, SHIMAZAKI Kei, NAGASAWA Junki, TSUCHIDA Sayaka, USHIDA Kazunari, MATSUBAYASHI Makoto, FURUYAMA Yuuki, OHGANE Kenji, KURAMOCHI Kouji, 原著, 研究論文(学術雑誌), 共著者
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Conversion of a PROTAC Mutant Huntingtin Degrader into Small-Molecule Hydrophobic Tags Focusing on Drug-like Properties
ACS Medicinal Chemistry Letters, , 2022年02月, HIRAI Keigo, YAMASHITA Hiroko, TOMOSHIGE Shusuke, MISHIMA Yugo, NIWA Tatsuya, OHGANE Kenji, ISHII Mayumi, KANAMITSU Kayoko, IKEMI Yui, NAKAGAWA Shinsaku, TAGUCHI Hideki, SATO Shinichi, HASHIMOTO Yuichi, ISHIKAWA Minoru, 原著, 研究論文(学術雑誌), 共著者
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Synthesis and Antiviral Activities of Neoechinulin B and Its Derivatives
Journal of Natural Products, , 85巻1号(頁284 - 291), 2022年01月, NISHIUCHI Kota, OHASHI Hirofumi, NISHIOKA Kazane, YAMASAKI Masako, FURUTA Masateru, MASHIKOTakumi, TOMOSHIGE Shusuke, OHGANE Kenji, KAMISUKI Shinji, WATASHI Koichi, KURAMOCHI Kouji, 原著, 研究論文(学術雑誌), 共著者
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Deoxygenation of tertiary and secondary alcohols with sodium borohydride, trimethylsilyl chloride, and potassium iodide in acetonitrile
Tetrahedron Letters, , 86巻(頁153519), 2021年12月, KATO Yuichi, INOUE Tomoka, FURUYAMA Yuuki, OHGANE Kenji, SADAIE Mahito, KURAMOCHI Kouji, 原著, 研究論文(学術雑誌), 共著者
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Deuteration of terminal alkynes realizes simultaneous live cell Raman imaging of similar alkyne-tagged biomolecules
Organic & Biomolecular Chemistry, , 2021年09月, Syusuke Egoshi, Kosuke Dodo, Kenji Ohgane, Mikiko Sodeoka, 原著, 研究論文(学術雑誌), 共著者
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Epo-C12 inhibits peroxiredoxin 1 peroxidase activity
Bioorganic & Medicinal Chemistry, , 41巻(頁116203 - ), 2021年07月, Tomoka Yoda, Masateru Furuta, Tomohiko Tsutsumi, Seiki Ikeda, Shunsuke Yukizawa, Satoshi Arai, Akinori Morita, Kenji Yamatoya, Kazuya Nakata, Shusuke Tomoshige, Kenji Ohgane, Yuuki Furuyama, Kengo Sakaguchi, Fumio Sugawara, Susumu Kobayashi, Masahiko Ikekita, Kouji Kuramochi, 原著, 研究論文(学術雑誌), 共著者
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SYNTHESIS, PHOTOCHEMICAL PROPERTIES, AND CYTOTOXICITY OF 10-ALKYLPHENAZIN-2(10H)-ONES
Heterocycles, , 102巻5号(頁871 - 885), 2021年05月, KOHATSU Haruki, KAMO Shogo, HOSOKAI Takuya, KAMISUKI Shinji, MACHIDA Yutaro, KOBAYASHI Ryota, KAWASAKI Tsuneomi, OHGANE Kenji, KURAMOCHI Kouji, 原著, 研究論文(学術雑誌), 共著者
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Image-based screen capturing misfolding status of Niemann-Pick type C1 identifies potential candidates for chaperone drugs
PLOS ONE, , 15巻12号(頁e0243746 - ), 2020年12月, Ryuta Shioi, Fumika Karaki, Hiromasa Yoshioka, Tomomi Noguchi-Yachide, Minoru Ishikawa, Kosuke Dodo, Yuichi Hashimoto, Mikiko Sodeoka, Kenji Ohgane, 原著, 研究論文(学術雑誌), 第一著者相当
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Bisphosphonate esters interact with HMG-CoA reductase membrane domain to induce its degradation
Bioorganic & Medicinal Chemistry, , 28巻14号(頁115576 - ), 2020年05月, Yosuke Toyota, Hiromasa Yoshioka, Ikuya Sagimori, Yuichi Hashimoto, Kenji Ohgane, 原著, 研究論文(学術雑誌), 第一著者相当